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6-bromo-3-(5,6-dimethoxy-3-pyridinyl)imidazo[1,2-a]pyridine
6-benzyl-3-iodoimidazo[1,2-c]pyrimidin-5(6H)-one
3-(5,6-dimethoxy-3-pyridinyl)imidazo[1,2-a]pyridine
6-benzylimidazo[1,2-c]pyrimidin-5(6H)-one
6-(pyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxylic acid
3-(6-methylpyridin-3-yl)-6-(pyridin-3-yl)imidazo[1,2-a]pyridine
3-bromo-7-methyl-6-(6-methylpyridin-3-yl)imidazo[1,2-a]pyridine
7-methyl-6-(6-methylpyridin-3-yl)imidazo[1,2-a]pyridine
3-bromo-6-(pyridin-3-yl)imidazo[1,2-a]pyridine
3-bromo-5,7-dimethyl-6-(pyridin-3-yl)imidazo[1,2-a]pyridine
5,7-dimethyl-6-(pyridin-3-yl)imidazo[1,2-a]pyridine
6-bromo-5,7-dimethylimidazo[1,2-a]pyridine
3-bromo-6-(6-methoxypyridin-3-yl)imidazo[1,2-a]pyridine
6-(6-methoxypyridin-3-yl)imidazo[1,2-a]pyridine
6-(pyridin-3-yl)imidazo[1,2-a]pyridine
5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzo[d]oxazol-2-amine
6-(4-(pyridin-4-yl)quinolin-6-yl)benzo[d]thiazol-2-amine
5-(3-(pyridin-4-yl)imidazo[1,2-a]pyridin-6-yl)benzo[d]oxazol-2-amine
2-acetamidobenzo[d]thiazol-6-ylboronic acid
tert-butyl 4-(7-(4-methanesulfonylphenyl)thieno[3,2-d]pyrimidin-4-yloxy)piperidin-1-carboxylate
4-(3-cyclohexyl-[1,2,4]oxadiazol-5-yl)piperidine
4-(3-cyclopentyl-[1,2,4]oxadiazol-5-yl)piperidine
tert-butyl 4-(3-cyclopropyl[1,2,4]oxadiazol-5-yl)piperidine-1-carboxylate
1-(5-isopropyl[1,2,4]oxadizol-3-yl)piperidin-4-ol
4,4,5,5-tetramethyl-2-[4-(propane-1-sulfonyl)phenyl][1,3,2]dioxaborolane
7-(4-methanesulfonylphenyl)-N-(piperidin-4-yl)thieno[3,2-d]pyrimidin-4-amine
tert-butyl 4-(7-bromothieno[3,2-d]pyrimidin-4-yloxy)piperidine-1-carboxylate
4-(methanesulfonyl)-7-(4-methanesulfonyl-phenyl)thieno[3,2-d]pyrimidine
7-(4-methanesulfonylphenyl)-4-methylsulfanylthieno[3,2-d]pyrimidine
1-(4-isopropylthiazo-2-yl)piperidin-4-ol
1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)pyrrolidin-3-ol
4-hydroxypiperidine-1-carboxylic acid tert-butylamide
7-bromo-4-chloro-5-ethyl-5H-pyrrolo[3,2-d]pyrimidine
4,N-dihydroxypiperidin-1-carboxamidine
1-iodo-4-(propane-1-sulfonyl)benzene
4-(3-cyclopropyl[1,2,4]oxadiazol-5-yl)piperidine
(S)-2-(methoxy-methyl-carbamoyl)-pyrrolidine-1-carboxylic acid tert-butyl ester
5-oxo-1-(3-phenoxyphenyl)-4,5-dihydro-1H-pyrazole-3-carboxylic acid
1-(2-acetylamino-phenyl)-5-oxo-4,5-dihydro-1H-pyrazole-3-carboxylic acid
1-([t-butyl(dimethyl)silyl]oxy)indane-5-carbaldehyde
4-methyl-5-oxo-1-vinyl-4,5-dihydro-1H-pyrazole-3-carboxylic acid methyl ester
4-methyl-5-oxo-1-vinyl-4,5-dihydro-1H-pyrazole-3-carboxylic acid
ethyl 4-(2-methyl-1-imidazolyl)benzoate
(N-cyclopropyl)-4-oxazol-5-yl-(N-piperidin-4-yl)benzamide
3-fluoro-4-(1H-1,2,4-triazol-1-yl)benzoic acid
4-(2-methyl-1H-imidazol-1-yl)benzoic acid
4-{cyclopropyl-[4-(4-methyl-oxazol-5-yl)-benzoyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester
N-cyclopropyl-4-oxazol-5-yl-N-(1-pyrimidin-2-ylpiperidin-4-yl)benzamide
N-cyclopropyl-4-oxazol-5-yl-N-(1-pyridin-2-ylpiperidin-4-yl)benzamide
N-cyclopropyl N-(3-methylpiperidin-4-yl)-4-oxazol-5-ylbenzamide
3-fluoro-4-(2-methyl-1H-imidazol-1-yl)benzoic acid
3-fluoro-4-(5-methyl-1H-1,2,4-triazol-1-yl)benzoic acid
3-fluoro-4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoic acid
3-Fluoro-4-(1H-1,2,3,4-tetrazol-1-yl)benzoic acid
4-(4-methyloxazol-5-yl)benzoyl chloride
4-(5-methyl-1H-1,2,4-triazol-1-yl)benzoic acid
N-hydroxy-but-3-enamidine
N-hydroxy-2-(tetrahydro-pyran-4-yl)acetamidine
4-(6-chloro-5-methyl-pyrimidin-4-ylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester
4-(6-chloro-5-methyl-pyrimidin-4-ylsulfanyl)-piperidine-1-carboxylic acid isopropyl ester
4-(2-chloro-3-methyl-pyridin-4-yloxy)-piperidine-1-carboxylic acid isopropyl ester
2-fluoro-4-(2-morpholin-4-yl-ethyl)-phenol
2-(4-benzyloxy-3-fluoro-phenyl)-ethanol
1-benzyloxy-4-(2-bromoethyl)-2-fluorobenzene
4-chloro-5-methyl-6-(piperidin-4-ylsulfanyl)-pyrimidine
1-methylethyl 4-({1-[4-(methylsulfonyl)phenyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
1-methylethyl 4-[(7-{4-[(dimethylamino)sulfonyl]phenyl}-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]-1-piperidinecarboxylate
1,1-dimethylethyl 4-[(1-{4-[(ethyloxy)carbonyl]phenyl}-2,3-dihydro-1H-indol-4-yl)oxy]-1-piperidinecarboxylate
1,1-dimethylethyl 4-[(1-{4-[(methylamino)carbonyl]phenyl}-2,3-dihydro-1H-indol-4-yl)oxy]-1-piperidinecarboxylate
1,1-dimethylethyl 4-({1-[5-(methylsulfonyl)-2-pyrimidinyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
4-{4-[(1-{[(1,1-dimethylethyl)oxy]carbonyl}-4-piperidinyl)oxy]-2,3-dihydro-1H-indol-1-yl}benzoic acid
1-methylethyl 4-({1-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
1-methylethyl 4-({1-[4-(1,3-thiazol-2-yl)phenyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
1-methylethyl 4-({1-[5-(methylsulfonyl)-2-pyrimidinyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
1-methylethyl 4-({1-[4-(3-furanyl)phenyl]-2,3-dihydro-1H-indol-4-yl}oxy)-1-piperidinecarboxylate
1-methylethyl 4-{[7-(4-bromophenyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl]oxy}-1-piperidinecarboxylate
1,1-dimethylethyl 4-{[1-(4-iodophenyl)-1H-indol-4-yl]oxy}-1-piperidinecarboxylate
4-(4-chloro-5,6-dihydro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-N,N-dimethylbenzenesulfonamide
2-{4-[(4-bromophenyl)amino]-6-chloro-5-pyrimidinyl}ethanol
N-[2-(4,6-dichloro-5-pyrimidinyl)ethyl]-5-fluoro-2-pyridinamine
1-methylethyl 4-[{[(1,1-dimethylethyl)oxy]carbonyl}(methyl)amino]-1-piperidinecarboxylate
N-[2-(4,6-dichloro-5-pyrimidinyl)ethyl]-2-methyl-3-pyridinamine
N-(4-bromophenyl)-6-chloro-5-(2-propen-1-yl)-4-pyrimidinamine
7-(4-bromophenyl)-4-chloro-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine
4-chloro-7-(2-methyl-3-pyridinyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidine
1-(5-fluoro-2-pyrimidinyl)-4-piperidinol
isopropyl 4-bromopiperidine-1-carboxylate
1,1-dimethylethyl 4-[(1-{4-[(ethyloxy)carbonyl]phenyl}-1H-indol-4-yl)oxy]-1-piperidinecarboxylate
1,1-dimethylethyl 4-{[1-(5-bromo-2-pyrimidinyl)-2,3-dihydro-1H-indol-4-yl]oxy}-1-piperidinecarboxylate
4-{[6-chloro-5-(2-propen-1-yl)-4-pyrimidinyl]amino}-2,5-difluorobenzonitrile
4-isopentyloxyphenol
6-butylsulfanylpyridin-3-ol
3-[4-(3-methylbutoxy)phenoxy]pyrrolidin-2-one
3-bromo-2-(cyclopropylmethoxy)-5-iodopyridine
5-bromo-6-(cyclopropylmethoxy)pyridin-3-ol
2-bromo-5-(4-methoxybenzyloxy)pyridine
6-ethoxy-5-fluoropyridin-3-ol
N-butyl-5-hydroxy-N-methylpyridine-2-carboxamide
(5-hydroxypyridin-2-yl)-pyrrolidin-1-yl-methanone
5-hydroxypyridine-2-carboxylic acid cyclopropylmethyl ester
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