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 6-(3-isopropyl-[1,2,4]oxadiazol-5-yl)pyridin-3-ol 2-(5-(4-methoxybenzyloxy)pyridin-2-yl)-5-methylthiazole 6-(5-methylthiazol-2-yl)pyridin-3-ol 6-(2-cyclopropylethoxy)pyridin-3-ol
 (1-(trifluoromethyl)cyclopropyl)methyl methanesulfonate methyl 4-(acetylamino)benzoate 3-(4-cyano-2-fluorophenyl)isoxazole-5-carboxylic acid 1-(5-methylpyrimidin-2-yl)piperidin-4-ol
 4-[(2-chloro-pyrimidine-5-carbonyl)-cyclopropyl-amino]-piperidine-1-carboxylic acid tert-butyl ester 5-(1H-1,2,4-triazol-1-yl)pyrazine-2-carboxylic acid 1-(5-methylpyrazin-2-yl)piperidin-4-ol 6-oxazol-5-yl-nicotinic acid
 4-{cyclopropyl-[6-(4-methanesulfonyl-phenyl)-pyridine-3-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester 4-{cyclopropyl-[2-(4-methanesulfonyl-phenyl)-pyrimidine-5-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester N-cyclopropyl-6-(4-methanesulfonyl-phenyl)-N-piperidin-4-yl-nicotinamide N-cyclopropyl-2-(4-(methylsulfonyl)phenyl)-N-(piperidin-4-yl)pyrimidine-5-carboxamide
 2-(4-(cyanomethyl)phenyl)-N-(1-cyclopropylpiperidin-4-yl)pyrimidine-5-carboxamide 4-[cyclopropyl-(2-imidazol-1-yl-pyrimidine-5-carbonyl)-amino]-piperidine-1-carboxylic acid tert-butyl ester 4-[(6-bromo-pyridine-3-carbonyl)-cyclopropyl-amino]-piperidine-1-carboxylic acid tert-butyl ester N-cyclopropyl-2-(1H-imidazol-1-yl)-N-(piperidin-4-yl)pyrimidine-5-carboxamide
 5-(3-methyl-1H-1,2,4-triazol-1-yl)pyrazine-2-carboxylic acid 5-(2-methyl-1H-imidazol-1-yl)pyrazine-2-carboxylic acid 6-(5-methyl-1H-1,2,4-triazol-1-yl)pyridine-3-carboxylic acid 2-(2-methyl-1H-imidazol-1-yl)pyrimidine-5-carboxylic acid
 6-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)pyridine-3-carboxylic acid 8-(3-phenyl-[1,2,4]oxadiazol-5-yl)-1,4-dioxa-8-aza-spiro[4.5]decane N-cyclopropyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-amine 1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-cyclopropylpiperidin-4-amine
 8-(3-propyl-[1,2,4]oxadiazol-5-yl)-1,4-dioxa-8-aza-spiro[4.5]decane 8-(3-tert-butyl-[1,2,4]oxadiazol-5-yl)-1,4-dioxa-8-aza-spiro[4.5]decane N-cyclopropyl-1-(3-isopropyl-1,2,4-oxadiazol-5-yl)piperidin-4-amine 8-(5-ethylpyrimidin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane
 N-cyclopropyl-1-(5-ethylpyrazin-2-yl)piperidin-4-amine 1-(5-chloropyrimidin-2-yl)-N-cyclopropylpiperidin-4-amine N-cyclopropyl-1-(5-ethylpyrimidin-2-yl)piperidin-4-amine 8-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-1,4-dioxa-8-aza-spiro[4.5]decane
 N-cyclopropyl-1-(5-methylpyrazin-2-yl)piperidin-4-amine 8-(5-chloropyrimidin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane 1-(3-phenyl-[1,2,4]oxadiazol-5-yl)piperidin-4-one N-cyclopropyl-1-(5-methylpyrimidin-2-yl)piperidin-4-amine
 1-(3-propyl-[1,2,4]oxadiazol-5-yl)-1,4-dioxa-8-aza-spiro[4.5]decane 1-(3-tert-butyl-[1,2,4]oxadiazol-5-yl)piperidin-4-one 1-(5-ethylpyrazin-2-yl)piperidin-4-ol 1-(5-ethylpyrazin-2-yl)piperidin-4-one
 1-(5-chloropyrimidin-2-yl)piperidin-4-one 1-(5-methylpyrazin-2-yl)piperidin-4-one 1-(5-methylpyrimidin-2-yl)piperidin-4-one 1,4-dioxa-8-aza-spiro[4.5]decane-8-carbonitrile
 2-bromo-5-ethylpyrazine 6-(2-methyl-1H-imidazol-1-yl)pyridine-3-carboxylic acid 1-(2-fluoro-4-methanesulfonylphenyl)-2-methyl-1H-imidazole-4-carboxylic acid 1-(2-fluoro-4-methanesulfonylphenyl)-1H-imidazole-4-carboxylic acid
 1-(4-cyano-2-fluorophenyl)-2-methyl-1H-imidazole-4-carboxylic acid 1-(5-cyanopyridin-2-yl)-2-methyl-1H-imidazole-4-carboxylic acid 1-(5-cyanopyridin-2-yl)-1H-imidazole-4-carboxylic acid 2-(5-methyl-1H-1,2,4-triazol-1-yl)pyrimidine-5-carboxylic acid
 5-oxazol-5-yl-pyrazine-2-carboxylic acid 2-(1H-1,2,4-triazol-1-yl)pyrimidine-5-carboxylic acid 2-imidazol-1-yl-pyrimidine-5-carboxylic acid methyl 1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazole-4-carboxylate
 5-(2-hydroxypropan-2-yl)-1H-pyrazole-3-carboxylic acid 4-amino-2-chloro-6-fluorobenzonitrile ethyl 5,7-dimethylimidazo[1,2-c]pyrimidine-2-carboxylate 4-bromo-3-chloro-5-fluoroaniline
 3-(ethoxycarbonyl)isoxazole-5-carboxylic acid Methyl-2-bromo-1-((2-(trimethylsilyl)ethoxy)methyl)-1H-imidazole-4-carboxylate 5,7-dimethylimidazo[1,2-c]pyrimidine-2-carboxylic acid 1-cyclopropyl-1H-pyrazole-3-carboxylic acid
 Methyl 1-cyclopropyl-1H-pyrazole-3-carboxylate 2-Chloro-6-fluoro-4-(1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl)benzonitrile 2-Chloro-4-(1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl)benzonitrile 2-Chloro-6-fluoro-4-iodobenzonitrile
 methyl 2-formyl-1-((2-(trimethylsilyl)-ethoxy)-methyl)-1H-imidazole-4-carboxylate 6-(methylsulfonamido)imidazo[1,2-a]pyridine-2-carboxylic acid Ethyl 5-(cyclopropylcarbamoyl)isoxazole-3-carboxylate Ethyl 5-(1,5-dimethyl-1H-pyrazol-3-yl)-1,2,4-oxadiazole-3-carboxylate
 Ethyl 7-oxo-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxylate 5-(cyclopropylcarbamoyl)isoxazole-3-carboxylic acid tert-butyl 5-(pyridin-3-yl)pyridine-2-carboxylate benzyl 2-bromo-1-methyl-1H-imidazole-4-carboxylate
 5-(1,5-dimethyl-1H-pyrazol-3-yl)-1,2,4-oxadiazole-3-carboxylic acid ethyl 5-oxo-5,6-dihydroimidazo[1,2-c]pyrimidine-2-carboxylate Ethyl 3-(1H-imidazol-4-yl)-1H-pyrazole-5-carboxylate ethyl 3-(1H-pyrazol-5-yl)-1H-pyrazole-5-carboxylate
 7-Oxo-5,6,7,8-tetrahydroimidazo[1,2-a]pyrimidine-2-carboxylic acid ethyl 2-(2-ethoxypropan-2-yl)oxazole-4-carboxylate 3-(1H-pyrazol-5-yl)-1H-pyrazole-5-carboxylic acid 1-methyl-2-(1-methyl-1H-pyrazol-4-yl)-1H-imidazole-4-carboxylic acid
 ethyl 5-(2-hydroxypropyl)-1H-pyrazole-3-carboxylate methyl 2-butyl-1-methyl-1H-imidazole-4-carboxylate 5-Oxo-5,6-dihydroimidazo[1,2-c]pyrimidine-2-carboxylic acid Ethyl 1,6-dihydropyrrolo[2,3-c]pyrazole-5-carboxylate
 2-chloro-4-(1H-pyrazol-3-yl)benzonitrile 6-Cyanoimidazo[1,2-a]pyridine-2-carboxylic acid Ethyl 5-(2-hydroxypropan-2-yl)-1H-pyrazole-3-carboxylate 5-(pyridin-3-yl)pyridine-2-carboxylic acid
 Ethyl 5-(1-hydroxy-2-methylpropyl)isoxazole-3-carboxylate ethyl 5-(isoxazol-3-yl)-1,2,4-oxadiazole-3-carboxylate methyl 2-butyl-1H-imidazole-4-carboxylate 2-cyclopropyl-1-methyl-1H-imidazole-4-carboxylic acid
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