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 3-ethynyl-4-methylbenzoyl chloride 4-amino-2-(trifluoromethyl)benzaldehyde 4-methyl-N-(3-pyridylmethyleneamino)benzenesulfonamide 3-cyano-4-methylbenzoic acid
 1-bromo-4-(cyclopentyloxy)benzene Ethyl 5-bromo-3-methylindole-2-carboxylate 4-cyclopentyloxy-phenylboronic acid 5-bromo-3-chloro-indole-2-carboxylic acid ethyl ester
 5-bromo-3-iodo-1H-indole-2-carboxylic acid ethyl ester 5-(4-tert-butylphenyl)indole-2-carboxylic acid ethyl ester 5-bromo-1H-indole-2-carboxamide 5-benzyloxy-1-(4-isopropoxyphenyl)indole-2-carboxylic acid ethyl ester
 5-hydroxy-1-(4-isopropoxyphenyl)indole-2-carboxylic acid ethyl ester 5-(5-trifluoromethylpyrid-2-yl)-1H-indole-2-carboxylic acid ethyl ester 5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1H-indole-2-carboxylic acid ethyl ester ethyl 5-(2-chloroacetyl)-1H-indole-2-carboxylate
 5-(1-tert-butoxycarbonyl-piperidin-4-yl)-1H-indole-2-carboxylic acid 5-(1-tert-butoxycarbonyl-piperidin-4-yl)-1H-indole-2-carboxylic acid ethyl ester 5-pyridin-3-yl-1H-indole-2-carboxylic acid ethyl ester 5-pyridin-4-yl-1H-indole-2-carboxylic acid ethyl ester
 5-(1-methylpyrrolidin-3-yl)-1H-indole N-(3-fluorophenyl)-5-(piperidin-3-yl)-1H-indole-2-carboxamide N-(3-fluorophenyl)-5-(1-((tetrahydrofuran-2-yl)methyl)piperidin-3-yl)-1H-indole-2-carboxamide ethyl 5-(1-(pyrrolidin-1-yl)propan-2-yl)-1H-indole-2-carboxylate
 ethyl 5-(3-(pyrrolidin-1-yl)prop-1-en-2-yl)-1H-indole-2-carboxylate ethyl 5-(2-(pyrrolidin-1-yl)acetyl)-1H-indole-2-carboxylate ethyl 5-(4-(piperidin-1-yl)but-1-en-2-yl)-1H-indole-2-carboxylate ethyl 5-(3-(piperidin-1-yl)propanoyl)-1H-indole-2-carboxylate
 ethyl 5-(1-(1-benzylpyrrolidin-3-yl)vinyl)-1H-indole-2-carboxylate 1-benzylpyrrolidine-3-carbonyl chloride ethyl 5-(1-benzylpyrrolidine-3-carbonyl)-1H-indole-2-carboxylate 5-(1-pyrrolidin-1-yl-ethyl)-1H-indole-2-carboxylic acid
 5-(1-pyrrolidin-1-yl-ethyl)-1H-indole-2-carboxylic acid ethyl ester 5-[1-(2-oxopiperidin-1-yl)ethyl]-1H-indole-2-carboxylic acid ethyl ester 5-[1-(2-oxopiperidin-1-yl)vinyl]-1H-indole-2-carboxylic acid ethyl ester 5-[1-(2-oxopyrrolidin-1-yl)ethyl]-1H-indole-2-carboxylic acid ethyl ester
 5-[1-(2-oxopyrrolidin-1-yl)vinyl]-1H-indole-2-carboxylic acid ethyl ester 5-bromo-1-(4-methoxybenzyl)-1H-indole-2-carboxylic acid ethyl ester 5-(4-isopropylpiperazin-1-yl)-1H-indole-2-carboxylic acid ethyl ester 1-isopropyl-4-(3-methyl-4-nitrophenyl)piperazine
 5-[1-(2-methoxy-ethyl)-piperidin-3-yl]-1H-indole-2-carboxylic acid ethyl ester 5-(1-methyl-piperidin-3-yl)-1H-indole-2-carboxylic acid ethyl ester 5-(1-methanesulfonyl-piperidin-3-yl)-1H-indole-2-carboxylic acid ethyl ester 5-piperidin-3-yl-1H-indole-2-carboxylic acid ethyl ester
 5-(1-isopropyl-piperidin-4-yl)-1H-indole-2-carboxylic acid hydrochloride N-(3-fluorophenyl)-5-(pyridin-3-yl)-1H-indole-2-carboxamide 5-piperidin-4-yl-1H-indole-2-carboxylic acid ethyl ester 5-(1-isopropyl-piperidin-3-yl)-1H-indole-2-carboxylic acid ethyl ester
 5-(1-isopropyl-piperidin-4-yl)-1H-indole-2-carboxylic acid ethyl ester 5-(3-ethyl-2,6-dioxo-piperidin-3-yl)-1H-indole-2-carboxylic acid 5-(3-isopropyl-5-oxo-pyrrolidin-3-yl)-1H-indole-2-carboxylic acid 4-(4-aminophenyl)-4-isopropylpyrrolidin-2-one
 4-(4-amino-3-iodophenyl)-4-isopropylpyrrolidin-2-one 5-(1-methyl-pyrrolidin-3-yl)-1H-indole-2-carboxylic acid 5-(1-benzyl-pyrrolidin-3-yl)-1H-indole-2-carboxylic acid 5-(1-benzyl-pyrrolidin-3-yl)-1H-indole
 2-(4-(piperazin-1-yl)phenyl)quinazolin-4(3H)-one N-(1-(4-formylphenyl)piperidin-4-yl)benzamide ethyl 4-(4-benzamidopiperidin-1-yl)benzoate N-(1-(4-formylphenyl)piperidin-4-yl)acetamide
 N-(1-(4-(hydroxymethyl)phenyl)piperidin-4-yl)acetamide ethyl 4-(4-acetamidopiperidin-1-yl)benzoate ethyl 4-(4-(methylsulfonyloxy)piperidin-1-yl)benzoate 2-(4-(3-aminopyrrolidin-1-yl)phenyl)-5,7-dimethoxyquinazolin-4(3H)-one
 2-(4-bromophenyl)-5,7-dimethoxyquinazolin-4(3H)-one 3-methyl-3-cyclobutyl-1-propyn-3-ol 4-(5-bromo-1-(2-methoxyethyl)-1H-indol-3-yl)pyrimidin-2-amine 5-iodo-4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine
 4-(6-bromo-4-(2-methoxyethoxy)-1H-indol-1-yl)pyrimidin-2-amine N-(1-(2-aminopyrimidin-4-yl)-6-bromo-1H-indol-4-yl)acetamide 5-chloro-4-(6-iodo-3,3-dimethyl-2,3-dihydro-1H-indol-1-yl)-2-pyrimidinamine 3-acetyl-5-bromo-N-cyclopropyl-1H-indole-2-carboxamide
 4-(5-iodo-1-(2-methoxyethyl)-1H-indol-3-yl)pyrimidin-2-amine 3-acetyl-5-bromo-N-(2-methoxyethyl)-1H-indole-2-carboxamide methyl 2-(4-bromo-2-nitrophenyl)-4-methylmorpholine-2-carboxylate 4-(5-bromo-1H-indol-3-yl)-5-chloro-N-methylpyrimidin-2-amine
 4-(5-bromo-1H-indol-3-yl)-5-chloropyrimidin-2-amine tert-butyl 6-bromo-3-hydroxymethyl-3-methyl-2,3-dihydro-1H-indole-1-carboxylate 2-(4-methyl-1-((4-methylphenyl)sulfonyl)-1H-imidazol-2-yl)-3-butyn-2-ol 1-(2-aminopyrimidin-4-yl)-6-bromo-1H-indol-4-ol
 4-(5-bromo-1H-indol-3-yl)-N-methylpyrimidin-2-amine 6-bromo-3-((2-methoxethoxy)methyl)-3-methyl-1,3-dihydro-2H-indol-2-one 4-(6-bromo-4-methoxy-1H-indol-1-yl)pyrimidin-2-amine tert-butyl 6-bromo-3-formyl-3-methyl-2,3-dihydro-1H-indole-1-carboxylate
 6-iodo-3,3-dimethyl-1-(1,3,5-triazin-2-yl)-2,3-dihydro-1H-indole dimethyl (4-bromo-2-nitrophenyl)(methyl)propanedioate 6-bromo-1-(2-chloropyrimidin-4-yl)indoline methyl (6-bromo-3-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetate
 6-bromo-3-((2-methoxethoxy)methyl)-3-methyl-2,3-dihydro-1H-indole 6-bromo-3,3-bis(hydroxymethyl)-1,3-dihydro-2H-indol-2-one 6-bromo-3-(3-hydroxypropyl)-3-methyl-1,3-dihydro-2H-indol-2-one 1-(4-methyl-1H-imidazol-2-yl)ethanone
 N-(6-bromoindolin-4-yl)acetamide 3-(6-bromo-3-methyl-2,3-dihydro-1H-indol-3-yl)-1-propanol methyl 6-bromo-3-methyl-2-oxo-2,3-dihydro-1H-indole-3-carboxylate methyl 2-(4-bromo-2-nitrophenyl)oxirane-2-carboxylate
 5-iodo-1-methyl-3-(pyrimidin-4-yl)-1H-indole 5-iodo-3-(isothiazol-5-yl)-1H-indazole 5-iodo-3-(pyrimidin-4-yl)-1H-indole 6-bromo-3-methyl-3-(2-propen-1-yl)-1,3-dihydro-2H-indol-2-one
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