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 2-(4-chloro-5-methyl-1H-pyrazol-3-yl)pyrimidine 2-(5-methyl-1(2)H-pyrazol-3-yl)-propan-2-ol 2-(4-iodo-pyrazol-1-yl)acetic acid ethyl 2-pyrrolo[2,3-b]pyridin-1-ylacetate
 ethyl 2-(3-iodo-1H-pyrazolo[3,4-b]pyridin-1-yl)acetate ethyl 3-(4-chloro-5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl)-2-methylpropanoate ethyl 2-(4-chloro-5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl)-2-methylpropanoate 4,5,6,7-tetrahydro-2H-pyrazolo[4,3-b]pyridine hydrochloride
 2-[5-methyl-3-(trifluoromethyl)-1,2,4-triazol-1-yl]propanoic acid 2-(4-chloro-5-methylpyrazol-1-yl)acetic acid 2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]propanoic acid 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethoxy)aniline
 methyl 5-bromoquinoline-8-carboxylate 5-bromo-1-methyl-1H-imidazol-2-amine 4-(3-fluorophenyl)-4-piperidinol 6-chloro-N-methylbenzo[d]thiazol-2-amine
 4-(2-chlorophenyl)-4-hydroxypiperidine 1,3-benzothiazole-4-sulfonyl chloride 4-(2-fluorobenzyl)piperidin-4-ol 4-isopropylpiperidin-4-ol
 1-tert-butyloxycarbonyl-4-(2-fluorobenzyl)-4-hydroxypiperidine tert-butyl 4-hydroxy-4-(2-methylallyl)piperidine-1-carboxylate tert-butyl 4-hydroxy-4-(pyridin-2-ylmethyl)piperidine-1-carboxylate (4-benzyl-piperidin-4-yl)methanol
 4-(ethoxymethyl)piperidin-4-ol 4-iodo-3-methylisothiazole methyl 4-(2-(benzyloxy)-2-oxoethoxy)-2-(diethoxymethyl)benzoate 2-(3-(diethoxymethyl)-4-(methoxycarbonyl)phenoxy)acetic acid
 (4-(tert-butyldimethylsilyloxy)-2-methylphenyl)(1H-imidazol-1-yl)methanone methyl 2-(diethoxymethyl)-4-hydroxybenzoate cyclopent-3-en-1-yl mesylate (2,6-dichloro-3-fluorophenyl)methanol
 4-bromo-5-chloro-1,3-dimethyl-1H-pyrazole 2-chloro-3-fluoro-6-methoxybenzaldehyde 4-bromo-3-methoxy-1-methyl-1H-pyrazole 1-(5,8-dioxaspiro[3.4]oct-2-yl)-5-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole
 5-bromo-1-(phenylsulfonyl)-2-(trimethylsilyl)-1H-pyrrolo[2,3-b]pyridine 1-[5-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-2-methylpropan-2-ol 1-[3-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-2-methylpropan-2-ol tert-butyl 4-(4-iodo-5-methyl-1H-pyrazol-1-yl)piperidine-1-carboxylate
 1-(1,4-dioxaspiro[4.5]dec-8-yl)-4-iodo-3,5-dimethyl-1H-pyrazole 1-(1,4-dioxaspiro[4.5]dec-8-yl)-4-iodo-3-methoxy-1H-pyrazole 1-(1,4-dioxaspiro[4.5]dec-8-yl)-3-ethyl-4-iodo-1H-pyrazole 1-(1,4-dioxaspiro[4.5]dec-8-yl)-4-iodo-3-methyl-1H-pyrazole
 1-(1,4-dioxaspiro[4.5]dec-8-yl)-4-iodo-5-methyl-1H-pyrazole 1-(cyclopent-3-en-1-yl)-4-iodo-3,5-dimethyl-1H-pyrazole 1-(4-iodo-3-methyl-1H-pyrazol-1-yl)-2-methylpropan-2-ol 1-(4-iodo-5-methyl-1H-pyrazol-1-yl)-2-methylpropan-2-ol
 1-(1-Methyl-1H-imidazol-2-yl)piperidin-4-ol 1-(Cyclopent-3-en-1-yl)-4-iodo-3-methyl-1H-pyrazole 1-(Cyclopent-3-en-1-yl)-4-iodo-5-methyl-1H-pyrazole 4-bromo-1-methyl-1H-pyrazole-3-carboxamide
 4-bromo-5-chloro-1-methyl-1H-pyrazole 4-bromo-3-chloro-1-methyl-1H-pyrazole 3-methoxy-1-methyl-1H-pyrazole 5-chloro-3,3-dimethyl-2,3-dihydroisoindol-1-one
 5-chloro-3-hydroxy-3-methyl-2,3-dihydroisoindol-1-one 1-(5-bromopyridin-3-ylmethyl)pyrrolidin-2-one ethyl 3-(3,5-dibromopyridin-4-yl)propanoate S)-1-(5-bromopyridin-3-ylmethyl)pyrrolidine-2-carboxylic acid methyl ester
 1-(5-bromo-pyridin-3-ylmethyl)-piperidin-2-one 1-(5-bromo-pyridin-3-yl)-pyrrolidin-2-one 3-bromo-5-(2-methylimidazol-1-ylmethyl)pyridine 5-chloro-2-(4-methoxybenzyl)-2,3-dihydroisoindol-1-one
 6-chloro-4-methyl-3,4-dihydro-2H-isoquinolin-1-one [2-(3-chlorophenyl)propyl]carbamic acid methyl ester N-(4-bromo-6,7-dihydro-5H-cyclopenta[c]pyridin-7-yl)acetamide 6-chloro-3-ethyl-3-hydroxy-2,3-dihydroisoindol-1-one
 N-(4-bromo-5,6,7,8-tetrahydroisoquinolin-8-yl)acetamide 3-bromo-5-(2-isopropylimidazol-1-ylmethyl)pyridine 6-chloro-3,3-dimethyl-2,3-dihydro-isoindol-1-one 1-(2-bromo-5-chlorophenyl)cyclopropanamine
 2-chloro-7,7-dimethyl-6,7-dihydropyrrolo[3,4-b]pyridin-5-one 5-chloro-3-cyclopropyl-2,3-dihydroisoindol-1-one 3-benzyl-5-chloro-2,3-dihydroisoindol-1-one [2-(3-chlorophenyl)-2-methylpropyl]carbamic acid methyl ester
 6-chloro-4,4-dimethyl-3,4-dihydro-2H-isoquinolin-1-one [2-(3-chlorophenyl)-1-methylethyl]carbamic acid methyl ester 8-chloro-3-methyl-3,4-dihydro-2H-isoquinolin-1-one 6-chloro-3-methyl-3,4-dihydro-2H-isoquinolin-1-one
 methyl 1,3-dimethyl-2-oxo-4-imidazolidinecarboxylate methyl 3-methyl-2-oxo-4-imidazolidinecarboxylate 1,1-dimethylethyl 1-methyl-2-oxo-4-imidazolidinecarboxylate tert-butyl 2-cyclohexyl-4,6-dioxopiperidine-1-carboxylate
 tert-butyl 2,4-dioxo-6-phenylpiperidine-1-carboxylate tert-butyl 2,4-dioxo-6-propylpiperidine-1-carboxylate tert-butyl 4-(3-phenylpropiolyl)piperazine-1-carboxylate (5-bromopyridin-3-yl)-(1-methyl-1H-imidazol-2-yl)methanol
 5-chloro-3-ethyl-3-hydroxy-2,3-dihydroisoindol-1-one 6-chloro-2-pyridin-3-yl-3,4-dihydro-2H-isoquinolin-1-one 3-bromo-5-(1-chloroethyl)pyridine ethyl 6-bromo-1,2-dihydro-4-hydroxy-2-oxoquinoline-3-carboxylate
 (4-amino-3-methylphenyl)(1-methyl-1H-imidazol-5-yl)methanone 5-(4-methylsulfonylbenzyl)-2,2-dimethyl-1,3-dioxane-4,6-dione 5-(4-(1H-pyrazol-1-yl)benzyl)-2,2-dimethyl-1,3-dioxane-4,6-dione 4-((6-bromo-4-chloro-2-methoxyquinolin-3-yl)methyl)benzonitrile
 4-((6-bromo-2,4-dichloroquinolin-3-yl)methyl)benzonitrile (2,4-dichloro-3-phenylquinolin-6-yl)(3,5-dimethylisoxazol-4-yl)methanol 2-(4-methylsulfonylbenzyl)malonic acid (2,4-dichloro-3-phenylquinolin-6-yl)(3-methylisoxazol-5-yl)methanone
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