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 4-[(furan-2-ylmethyl)-amino]-phthalic acid dimethyl ester 4-[(furan-2-ylmethyl)-amino]-phthalic acid 6-(2-oxo-oxazolidin-3-yl)-hexanoic acid ethyl ester 6-(2-oxo-oxazolidin-3-yl)-hexanoic acid
 5-(ethylthio)picolinic acid 3,4-Dihydro-3-trimethylsilyloxy-2H-pyran 1-bromo-4-(1-propylsulfonyl)benzene 1-bromo-3-(cyclopropylsulfanyl)benzene
 1-(3-bromophenyl)cyclopropanecarboxamide 2-(3-(cyclopropylsulfonyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-benzyl-6-bromo-3,4-dihydroisoquinolin-1(2H)-one 4-(4-fluorobenzoylamino)benzoyl chloride
 4-(3,4-dimethoxy-benzoylamino)-naphthalene-1-carboxylic acid ethyl ester 4-(3,4-dimethoxy-benzoylamino)-naphthalene-1-carbonyl chloride 4-(3,4-dimethoxy-benzoylamino)-naphthalene-1-carboxylic acid N-cyclohexylmethyl-N-4-nitrobenzamide
 6-amino-2-benzyl-3,4-dihydro-2H-isoquinolin-1-one N-isobutyl-3-nitroterephthalamic acid N-isobutyl-3-nitroterephthalamic acid methyl ester tert-butyl 4-(6-methoxy-1-oxo-3,4-dihydroisoquinolin-2(1H)-yl)piperidine-1-carboxylate
 2-(1-cyclobutylpiperidin-4-yl)-6-hydroxy-3,4-dihydroisoquinolin-1(2H)-one tert-butyl 4-(5-bromo-1-oxoisoindolin-2-yl)piperidine-1-carboxylate 6-hydroxy-2-(piperidin-4-yl)-3,4-dihydroisoquinolin-1(2H)-one methyl 5-acetyl-2-thiophenecarboxylate
 4-(1H-pyrazol-3-yl)benzonitrile 4-bromo-3-(4-chlorophenyl)-1H-pyrazole 2-(methylthio)-5-[tri(n-butyl)stannyl]thiophene 5-(1H-pyrazol-3-yl)-thiophene-2-carboxylic acid methyl ester
 6-bromo-8-methylimidazo[1,2-a]pyridine 6-bromo-4-(4-methylpiperazin-1-yl)quinoline 3-(dimethylamino)-2,2-dimethylpropan-1-ol 3-(1-benzyl-1H-1,2,3-triazol-4-yl)propan-1-ol
 N-allyl-2-bromobenzenesulfonamide 4-bromo-3-methyl-2-nitroaniline 6-bromo-2-methyl-1,2,3,4-tetrahydroisoquinoline 5-bromo-1-propyl-1,2-dihydropyridin-2-one
 1-methyl-5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1H-benzotriazole 2-bromo-N-(2-methylallyl)benzenesulfonamide N-benzyl-4-hydroxy-N-methylbutanamide N-methylcyclohexanesulfonamide
 (2-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)methanol methyl 3-(1-ethyl-1H-imidazol-4-yl)propanoate 4-bromo-3-chloro-N-methyl-2-nitroaniline 4-bromo-3-chloro-N1-methylbenzene-1,2-diamine
 5-bromo-N,4-dimethyl-3-nitropyridin-2-amine 2-(4-methoxybenzyl)isoindolin-1-one 5-bromo-2-cyclopropylisoindolin-1-one 2-methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3,4-dihydroisoquinolin-1(2H)-one
 6-chloro-3-iodo-1H-pyrazolo[3,4-b]pyridine ethyl 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-benzofuran-2-carboxylate 5-bromo-2-(2-(dimethylamino)ethyl)isoindolin-1-one 5-bromo-2-(2-methoxyethyl)isoindolin-1-one
 6-chloro-3-(1-methyl-1H-pyrazol-4-yl)-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-c]pyridine 6-chloro-3-iodo-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-c]pyridine 6-chloro-3-iodo-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-b]pyridine 6-(3,5-dimethoxyphenyl)-3-iodo-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-b]pyridine
 6-(3,5-dimethoxyphenyl)-3-iodo-1H-pyrazolo[4,3-b]pyridine 6-(3,5-dimethoxyphenyl)-1H-pyrazolo[4,3-b]pyridine 2-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 5-bromo-2-[2-(1-methylpyrrolidin-2-yl)ethyl]isoindolin-1-one
 2-[2-(dimethylamino)ethyl]-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 2-(1-methylpiperidin-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 5-bromo-2-(1-methylpiperidin-4-yl)isoindolin-1-one methyl 4-bromo-5-fluoro-2-methylbenzoate
 methyl 4-bromo-2-(bromomethyl)-5-fluorobenzoate 2-(2-hydroxypropyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 5-bromo-2-(2-hydroxypropyl)isoindolin-1-one 2-(2-hydroxy-1-methylethyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one
 2-(tetrahydro-2H-pyran-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 2-(2-methoxyethyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one (6-ethyl-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-3-yl)boronic acid 3-bromo-6-ethyl-5,6-dihydro-7H-pyrrolo[3,4-b]pyridin-7-one
 2-isopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 2-ethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-1-one 6-(3,5-dimethoxyphenyl)-3-iodo-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-c]pyridine 6-(3,5-dimethoxyphenyl)-3-iodo-1H-pyrazolo[4,3-c]pyridine
 6-(3,5-dimethoxyphenyl)-1H-pyrazolo[4,3-c]pyridine 2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]propanenitrile N,N-dimethyl-2-[2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]acetamide 2-(4-bromo-2-methylphenoxy)-N,N-dimethylacetamide
 6-(2,6-dichloro-3,5-dimethoxyphenyl)-3-iodo-1H-pyrazolo[4,3-c]pyridine 6-(2,6-dichloro-3,5-dimethoxyphenyl)-1H-pyrazolo[4,3-c]pyridine 6-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-c]pyridine 6-(3,5-dimethoxyphenyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[4,3-c]pyridine
 6-[6-(2,6-dichloro-3,5-dimethoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl]-3,4-dihydroisoquinolin-1(2H)-one 1-methyl-4-{[5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3-dihydro-1-benzofuran-2-yl]carbonyl}piperazine 1-[(5-bromo-2,3-dihydro-1-benzofuran-2-yl)carbonyl]-4-methylpiperazine N,N-dimethyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)chromane-2-carboxamide
 6-(2,6-dichloro-3,5-dimethoxyphenyl)-3-iodo-1H-pyrazolo[3,4-d]pyrimidine 6-(2,6-dichloro-3,5-dimethoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidine 6-(3,5-dimethoxyphenyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-d]pyrimidine 6-chloro-1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazolo[3,4-d]pyrimidine
 N,N-dimethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3-dihydro-1-benzofuran-2-carboxamide 5-bromo-N,N-dimethyl-2,3-dihydro-1-benzofuran-2-carboxamide 2-(chloromethyl)-5-(2-chloro-phenyl)-1,3,4-oxadiazole ethyl N-({2-[(4-chlorophenyl)carbonyl]hydrazinyl}carbonyl)glycinate
 [3-(4-chlorophenyl)-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl]acetic acid 2-methyl-5-(2-chlorophenyl)-1,3,4-thiadiazole 5-(4-chlorophenyl)-4-cyclopropyl-2,4-dihydro-3H-1,2,4-triazol-3-one 2-(chloromethyl)-5-(4-chlorophenyl)-4-cyclopropyl-2,4-dihydro-3H-1,2,4-triazol-3-one
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