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 6-chloropyrazine-2-carboxylic chloride 2-chloro-6-(trifluoromethyl)quinoxaline 5-amino-3-methyl-1,2-thiazole-4-carboxylic acid 5-amino-N-(3,4-dichlorophenyl)-3-methyl-1,2-thiazole-4-carboxamide
 5-amino-N-(6-methoxypyridin-3-yl)-3-methyl-1,2-thiazole-4-carboxamide 5-amino-N-(6-isopropoxypyridin-3-yl)-3-methyl-1,2-thiazole-4-carboxamide 2-chloro-6-(oxazol-2-yl)pyrazine 6-chloro-N-methylpyrazine-2-carboxamide
 2-chloro-6-(1H-pyrazol-1-yl)-pyrazine 2-chloro-N,N-dimethyl-1,3-thiazole-5-carboxamide 5-amino-N-(2-ethylphenyl)-3-methyl-1,2-thiazole-4-carboxamide N-(2-ethylphenyl)-3-methyl-5-(pyridin-2-ylamino)-1,2-thiazole-4-carboxamide
 5-amino-N-(6-ethoxypyridin-3-yl)-3-methyl-1,2-thiazole-4-carboxamide 6-chloro-N,N-dimethylpyrazine-2-carboxamide (2-chloro-1,3-thiazol-5-yl)(morpholin-4-yl)methanone 6-bromo-N-methylpyridazine-3-carboxamide
 6-chloro-N-ethylpyrazine-2-carboxamide methyl 4-nitrobiphenyl-2-carboxylate methyl 3-chloro-6-(trifluoromethyl)pyridine-2-carboxylate methyl 3-(pyrimidin-2-yl)-6-(trifluoromethyl)picolinate
 5-cyano-2-(pyrimidin-2-yl)benzoic acid methyl 5-cyano-2-(pyrimidin-2-yl)benzoate N,N-di-methyl-2-phenyl-5-aminobenzoic acid methyl N,N-di-methyl-2-phenyl-5-aminobenzoate
 methyl 2-phenyl-5-aminobenzoate 3-fluoro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2-methoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoic acid methyl ester 3-fluoro-2-(1H-1,2,3-triazol-1-yl)benzoic acid
 ethyl 2-bromo-6-methoxybenzoate 2-(methylsulfinyl)benzo[d]oxazole Methyl 3-bromo-6-methylpicolinate 4-[2-(5-bromo-2-chloro-pyridin-4-yl)-1-hydroxy-1-methyl-ethyl]-piperidine-1-carboxylic acid tert-butyl ester
 4-[2-(5-bromo-2-chloropyridin-4-yl)-1-hydroxy-ethyl]piperidine-1-carboxylic acid tert-butyl ester 4-[2-(5-bromo-2-chloropyridin-4-yl)acetyl]piperidine-1-carboxylic acid tert-butyl ester 4-(5-chloro-2-methyl-2,3-dihydrofuro[2,3-c]pyridin-2-yl)piperidine-1-carboxylic acid tert-butyl ester 4-(5-chloro-2,3-dihydrofuro[2,3-c]pyridin-2-yl)piperidine-1-carboxylic acid tert-butyl ester
 4-[5-(1-methanesulfonyl-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydrofuro[2,3-c]pyridin-2-yl]piperidine-1-carboxylic acid tert-butyl ester 4-[5-(4-methanesulfonylmethylphenyl)-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid tert-butyl ester 4-[5-(4-methanesulfonylphenyl)-2,3-dihydrofuro[2,3-c]pyridin-2-yl]-piperidine-1-carboxylic acid tert-butyl ester 4-[5-(4-methanesulfonylphenyl)furo[2,3-c]pyridin-2-yl]piperidine-1-carboxylic acid tert-butyl ester
 5-(1-methanesulfonyl-1,2,3,6-tetrahydropyridin-4-yl)-2-piperidin-4-yl-2,3-dihydrofuro[2,3-c]pyridine 5-(4-methanesulfonylmethylphenyl)-2-piperidin-4-yl-2,3-dihydrofuro[2,3-c]pyridine 5-(4-methanesulfonylphenyl)-2-piperidin-4-yl-2,3-dihydrofuro[2,3-c]pyridine 4-(5-chlorofuro[2,3-c]pyridin-2-yl)piperidine-1-carboxylic acid tert-butyl ester
 4-[5-(4-methanesulfonylphenyl)-2,3-dihydrobenzofuran-2-yl]piperidine 4-(5-bromo-2,3-dihydrobenzofuran-2-yl)piperidine-1-carboxylic acid tert-butyl ester 1-[4-(5-bromo-2,3-dihydrobenzofuran-2-yl)piperidin-1-yl]-2,2,2-trifluoroethanone 1-[4-(2,3-dihydrobenzofuran-2-yl)-piperidin-1-yl]-2,2,2-trifluoroethanone
 1-(4-benzofuran-2-yl-piperidin-1-yl)-2,2,2-trifluoroethanone 4-{2-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-2,3-dihydrobenzofuran-5-yl}benzoic acid 4-[5-(4-methanesulfonylphenyl)-2,3-dihydrobenzofuran-2-yl]piperidine-1-carbonitrile 4-(2-piperidin-4-yl-2,3-dihydro-benzofuran-5-yl)-benzoic acid methyl ester
 tert-butyl 4-{[1-(1-methylethyl)-4-piperidinyl]oxy}-1-piperidinecarboxylate 5-bromo-N-cyclobutylpicolinamide 4-{4-[(1-tert-butoxycarbonyl-4-piperidinyl)oxy]-1-piperidinyl}benzonitrile ethyl 6-[4-(4-piperidinyloxy)-1-piperidinyl]-3-pyridinecarboxylate
 tert-butyl 4-{[1-(cyclopropylmethyl)-4-piperidinyl]oxy}-1-piperidinecarboxylate tert-butyl 4-[(1-cyclobutyl-4-piperidinyl)oxy]-1-piperidinecarboxylate 1-cyclobutyl-4-(4-piperidinyloxy)piperidine 1-(cyclopropylmethyl)-4-(4-piperidinyloxy)piperidine
 1-isopropyl-4-(4-piperidinyloxy)piperidine 1-(4-{4-[(1-cyclobutyl-4-piperidinyl)oxy]-1-piperidinyl}phenyl)ethanone 5-(4-bromophenyl)-2-methyl-1,3-oxazole 1-(5-cyanopyridin-2-yl)piperidine-4-carboxylic acid
 ethyl 1-(5-cyano-pyridin-2-yl)-piperidine-4-carboxylate 1-isopropyl-4-(piperidine-4-carbonyl)-piperazine 5-(trifluoromethyl)-pyrazin-2(1H)-one 1-benzyl-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one
 1-(4-iodophenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4-ol 1-benzyl-3-chloro-5-methoxypyridazin-4(1H)-one 1-(1-benzyl-1H-pyrazol-4-yl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one
 1-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)propan-2-one 1-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-propan-2-ol 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-(1,3-thiazol-2-yl)pyridazin-4(1H)-one 1-(4-iodo-2-methoxyphenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one
 1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]pyridazin-4(1H)-one 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-(1,2,3,6-tetrahydropyridin-4-yl)pyridazin-4(1H)-one 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-piperidin-4-ylpyridazin-4(1H)-one
 5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)-1-pyridin-4-ylpyridazin-4(1H)-one 1-methoxy-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)propan-2-one 1-(dicyclopropylmethyl)-1H-pyrazol-4-amine 2-fluoro-4-(tetrahydro-2H-pyran-4-yl)aniline
 4-(3,6-dihydro-2H-pyran-4-yl)-2-fluoroaniline 1-(benzyloxy)-3-[(2-fluoro-4-iodophenyl)hydrazono]pentane-2,4-dione 3-acetyl-1-(4-iodo-2-methoxyphenyl)-5-methoxypyridazin-4(1H)-one 5-methoxy-2-methylisophthalic acid
 1-prop-2-ynyl-1H-indole-2-carboxylic acid methyl 1-(prop-2-ynyl)indole-2-carboxylate 1-(pyridin-4-yl)ethanamine dihydrochloride 1-(3-cyano-benzyl)-1H-indole-2-carboxylic acid ethyl ester
 1-(3-cyano-benzyl)-1H-indole-3-carboxylic acid 2,3,5-trichlorobenzylamine 2,3,5-trichlorophenylmethanol 1,4-dioxaspiro[4.5]decan-8-yl 4-methylbenzenesulfonate
 4-(4-bromophenyl)-4-(methoxymethyl)tetrahydro-2H-pyran tert-butyl 4-[4-(ethoxycarbonyl)benzylidene]piperidine-1-carboxylate tert-butyl 4-(4-cyanobenzylidene)piperidine-1-carboxylate {3-chloro-4-[(1-cyclobutylpiperidin-4-ylidene)methyl]phenyl}methanol
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