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 3-oxo-3-(tetrahydrofuran-3-yl)propanenitrile methyl 2,6-dimethylpyridine-4-carboxylate 3-cycloheptyl-3-oxo-propionitrile 4-chloro-3,3-dimethylbutane-2-one
 4-chloro-1-(4-chlorophenoxy)-3,3-dimethyl-butan-2-one 4-chloro-1-(4-chlorophenoxy)-3,3-dimethyl-1-(imidazol-1-yl)-butan-2-ol 1-bromo-4-chloro-1-(4-chlorophenoxy)-3,3-dimethyl-butan-2-one 4-chloro-1-[4-(4-chlorophenyl)-phenoxy]-3,3-dimethyl-butan-2-one
 4-chloro-1-(4-chloro-phenoxy)-3,3-dimethyl-1-[1,2,4]triazol-1-yl-butan-2-one 4-chloro-1-[4-(4-chlorophenyl)-phenoxy]-3,3-dimethyl-1-(1,2,4-triazol-1-yl)-butan-2-one 1-Phenazinamine 3-bromo-2-methyl-benzylamine hydrochloride
 methyl 2-(dichloromethyl)-1,3-oxazole-4-carboxylate ethyl 2-[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]-1,3-oxazole-4-carboxylate 2-[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]-1,3-oxazole-4-carboxylic acid 3-[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]propanoic acid
 {[3-bromo-2-(methyloxy)phenyl]methyl}amine hydrochloride methyl 2-{[bis(ethyloxy)phosphoryl]methyl}-1,3-oxazole-4-carboxylate diethyl 2-(1-chloroethylidene)malonate ethyl 6-ethyl-1-ethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate
 ethyl 1-ethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate [1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methanol 5-(aminomethyl)-1,6-diethyl-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine 1-ethyl-6-methyl-4-oxo-4,7-dihydro-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester
 ethyl 4-[(1-{[(1,1-dimethylethyl)oxy]carbonyl}-4-piperidinyl)amino]-1,6-diethyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylate [1-ethyl-6-methyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methanol [1-ethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methanol 5-(chloromethyl)-1-ethyl-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine
 4-{[5-(aminomethyl)-1,6-diethyl-1H-pyrazolo[3,4-b]pyridin-4-yl]amino}-1-piperidinecarboxamide 5-(aminomethyl)-1-ethyl-6-methyl-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine 5-(aminomethyl)-1-ethyl-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine ethyl 1-ethyl-6-methyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridine-5-carboxylat
 ethyl 1,6-diethyl-4-hydroxy-1H-pyrazolo[3,4-b]pyridine-5-carboxylate 4-nitro-N-isopropylphthalimide N-isopropyl-4-aminophthalimide 7-(4-chloro-benzylamino)-2-ethyl-4,4-dimethyl-3,4-dihydro-2H-isoquinolin-1-one
 5-(4-chloro-benzylamino)-2-isopropyl-isoindole-1,3-dione 7-(4-chloro-benzylamino)-4,4-dimethyl-3,4-dihydro-2H-isoquinolin-1-one 5-(4-chloro-benzylamino)-2-ethyl-2,3-dihydro-isoindol-1-one 6-benzylamino-3,4-dihydro-2H-isoquinolin-1-one
 2-bromo-N-ethyl-N-(2-methyl-allyl)-5-nitrobenzamide 2-ethyl-4,4-dimethyl-7-nitro-3,4-dihydro-2H-isoquinolin-1-one 7-amino-2-ethyl-4,4-dimethyl-3,4-dihydro-2H-isoquinolin-1-one 2-bromo-N-ethyl-5-nitro-benzamide
 2-ethyl-5-nitro-2,3-dihydro-isoindol-1-one 5-amino-2-ethyl-2,3-dihydro-isoindol-1-one 6-amino-2-ethyl-2,3-dihydro-isoindol-1-one 1-(4-(tert-butyl)phenyl)-3-chloropropan-1-one
 3-(4-phenylthiobenzoyl)propionic acid 6-chloro-2-methyl-4-({5-[(morpholin-4-yl)carbonyl]pyridin-2-yl}amino)-2,3-dihydropyridazin-3-one 7-phenylsulfanyl-3,4-dihydro-2H-naphthalen-1-one 6-cyclopropyl-3,4-dihydro-2H-isoquinolin-1-one
 6-dimethylamino-3,4-dihydro-2H-isoquinolin-1-one (3-bromo-2-methyl-phenyl)-acetic acid benzyl ester 7-benzenesulfonyl-3,4-dihydro-2H-naphthalen-1-one 6-Benzenesulfonyl-3,4-dihydro-2H-naphthalen-1-one
 6-phenylsulfanyl-3,4-dihydro-2H-naphthalen-1-one 3-(3-bromo-2-methylphenyl)-7-dimethylamino-1H-quinolin-4-one 6-tert-butyl-3,4-dihydroisoquinolin-1(2H)-one 6-(3-chloro-benzenesulfonyl)-3,4-dihydro-2H-naphthalen-1-one
 2-chloro-1-fluoro-4-(2-nitrovinyl)benzene 1-ethyl-1,4,5,6-tetrahydro-pyrrolo[2,3-c]pyridin-7-one N-[2-(3,4-dimethoxyphenyl)ethyl]carbamic acid ethyl ester 2-(4-chloro-3-methoxyphenyl)ethanamine
 3-(2-aminoethyl)-1-(4-methoxybenzyl)indole 3,4-dihydro-2,6-naphthyridin-1(2H)-one 2-(1-ethyl-1H-indol-3-yl)ethylamme 2-bromo-5-(2-nitrovinyl)thiophene
 1-chloro-2-fluoro-4-(2-nitrovinyl)benzene 5-fluorobenzo[b]thiophene-2-carboxaldehyde 2-(2-nitrovinyl)benzo[b]thiophene 7-(trifluoromethyl)-3,4-dihydroisoquinolin-1(2H)-one
 2-methyl-2-(4-trifluoromethylphenyl)propylamine 2-(4-methyl-pyridin-3-yl)-7-nitro-3,4-dihydro-2H-isoquinolin-1-one 3-(2-hydroxyethyl)-N-(4-methoxybenzyl)isonicotinamide 7-chloro-2-(4-ethylpyridin-3-yl)-3,4-dihydroisoquinolin-1(2H)-one
 7-amino-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 6-hydroxy-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 7-hydroxy-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 2-(4-methylpyridin-3-yl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-7-carbonitrile
 2-(4-methyl-pyridin-3-yl)-7-nitro-2H-isoquinolin-1-one 1-ethyl-6-(4-methyl-pyridin-3-yl)-1,4,5,6-tetrahydro-pyrrolo[2,3-c]pyridin-7-one 6-methyl-2-(4-methylpyridin-3-yl)-3,4-dihydroisoquinolin-1(2H)-one [2-(1-ethyl-1H-indol-3-yl)-1-methylethyl]carbamic acid ethyl ester
 5-Chloro-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one [2-(1-ethyl-1H-indol-3-yl)ethyl]carbamic acid ethyl ester 5-methoxy-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 2-(4-methoxybenzyl)-3,4-dihydro-2,6-naphthyridin-1(2H)-one
 6-methoxy-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 7-methoxy-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one ethyl 2-(5-fluorobenzo[b]thiophen-2-yl)ethylcarbamate ethyl 3-(3-chloro-4-(trifluoromethyl)phenyl)propanoate
 [2-(5-fluorobenzo[b]thiophen-3-yl)ethyl]carbamic acid ethyl ester 7-chloro-2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 7-amino-2-(4-methylpyridin-3-yl)-2H-isoquinolin-1-one 7-chloro-2-pyridin-3-yl-3,4-dihydro-2H-isoquinolin-1-one
 [2-(3-trifluoromethylphenyl)ethyl]carbamic acid ethyl ester [2-(4-trifluoromethylphenyl)ethyl]carbamic acid ethyl ester 7-(trifluoromethoxy)-3,4-dihydroisoquinolin-1(2H)-one [2-(2-trifluoromethylphenyl)ethyl]carbamic acid ethyl ester
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