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 2-(4-methylpyridin-3-yl)-3,4-dihydro-2,6-naphthyridin-1(2H)-one 2-(4-methyl-pyridin-3-yl)-3,4-dihydro-2H-isoquinolin-1-one 2-(4-methylpyridin-3-yl)-3,4-dihydro-2,7-naphthyridin-1(2H)-one 5-(4-methyl-pyridin-3-yl)-6,7-dihydro-5H-thieno[3,2-c]pyridin-4-one
 6-(4-methyl-pyridin-3-yl)-5,6-dihydro-4H-thieno[2,3-c]pyridin-7-one 6-trifluoromethyl-3,4-dihydro-2H-isoquinolin-1-one [2-(2-fluoro-5-methoxyphenyl)ethyl]carbamic acid ethyl ester [2-(4-chloro-3-fluorophenyl)ethyl]carbamic acid ethyl ester
 [2-(3-chloro-4-fluorophenyl)ethyl]carbamic acid ethyl ester 7-chloro-6-methoxy-3,4-dihydroisoquinolin-1(2H)-one 5-fluoro-8-methoxy-3,4-dihydro-2H-isoquinolin-1-one 5-pyridin-3-yl-6,7-dihydro-5H-thieno[3,2-c]pyridin-4-one
 6-pyridin-3-yl-5,6-dihydro-4H-thieno[2,3-c]pyridin-7-one 2-fluoro-4-(2-nitrovinyl)-1-trifluoromethylbenzene 1-ethyl-3-(2-nitro-propenyl)-1H-indole [2-(4-bromothiophen-2-yl)ethyl]carbamic acid ethyl ester
 [2-(5-bromothiophen-2-yl)ethyl]carbamic acid ethyl ester [2-(2-chlorophenyl)ethyl]carbamic acid ethyl ester 1-oxo-1,2,3,4-tetrahydro-isoquinoline-7-carbonitrile (E)-5-fluoro-2-(2-nitrovinyl)benzo[b]thiophene
 2-(1-ethyl-1H-indol-3-yl)-1-methylethylamine 2-bromo-6,7-dihydro-5H-thieno[3,2-c]pyridin-4-one 2-(5-fluorobenzo[b]thiophen-2-yl)ethanamine 3-bromo-6,7-dihydro-5H-thieno[3,2-c]pyridin-4-one
 1-ethyl-3-(2-nitro-vinyl)-1H-indole 3-(2-hydroxyethyl)isonicotinonitrile 4-(4-fluorophenylamino)-5,6-dihydropyridin-2(1H)-one 2-(5-fluorobenzo[b]thiophen-3-yl)ethylamine
 N-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-2-methoxy-6-methyl-phenyl]-3,3-dimethyl-butanamide N-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-2,6-dimethoxy-phenyl]-3,3-dimethyl-butanamide N-(4-(3,4-dihydroisoquinolin-2(1H)-yl)-2,6-dimethylphenyl)-3,3-dimethylbutanamide N-[2-Chloro-4-(3,4-dihydro-1H-isoquinolin-2-yl)-6-methyl-phenyl]-3,3-dimethyl-butanamide
 N-[2-chloro-4-(6-chloro-3,4-dihydro-1H-isoquinolin-2-yl)-6-methyl-phenyl]-3,3-dimethylbutanamide N-[4-(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-2,6-dimethyl-phenyl]-3,3-dimethylbutanamide N-[4-(6-chloro-3,4-dihydro-1H-isoquinolin-2-yl)-2,6-dimethyl-phenyl]-3,3-dimethylbutanamide (4-bromo-2-methoxy-6-methyl-phenyl)-3,3-dimethylbutanamide
 N-(4-Bromo-2,6-dimethoxy-phenyl)-3,3-dimethylbutanamide 2-allyl-4-chlorophenol (2-Naphthyl)oxamic acid ethyl ester 2-allyl-4-fluorophenol
 2-amino-7-methoxynaphthalene 4-(triisopropylsilyloxy)aniline 2,3-dihydro-2-(iodomethyl)benzofuran 1-(naphthalen-2-yl)piperazine hydrochloride
 2-chloromethyl-5-chlorobenzofuran 1-(allyloxy)-4-(trifluoromethyl)benzene 2-allyl-4-(trifluoromethyl)phenol (5-chloro-2,3-dihydro-1-benzofuran-2-yl)methanol
 (5-fluoro-2,3-dihydrobenzofuran-2-yl)methanol 2-chloro-1-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]ethan-1-one 5-fluoro-2,3-dihydro-benzofuran-2-carboxylic acid 2-chloromethyl-5-trifluoromethyl-benzoxazole
 (5-chloro-1-benzofuran-2-yl)methanamine 6-(trifluoromethyl)quinolin-2-amine tert-butyl 4-[[4-nitro-3-(trifluoromethyl)phenyl]amino]piperidine-1-carboxylate tert-butyl 4-(6-chloroquinolin-2-yl)piperazine-1-carboxylate
 4-[[4-nitro-3-(trifluoromethyl)phenyl]amino]phenol 5-fluoro-2-(piperazin-1-ylmethyl)-1,3-benzothiazole ethyl[[(5-chloro-1-benzofuran-2-yl)methyl]carbamoyl]formate 2-(azidomethyl)-5-chloro-1-benzofuran
 7-nitro-8-(trifluoromethyl)naphthalen-2-ol 7-methoxy-2-nitro-1-(trifluoromethyl)naphthalene 1-iodo-7-methoxy-2-nitronaphthalene 1-iodo-7-methoxynaphthalen-2-amine
 2-bromo-5-trifluoromethyl-benzothiazole 3-chloromethyl-7-trifluoromethyl-quinoline ethyl 2-oxo-2-(quinolin-2-ylamino)acetate 4-nitro-3-(trifluoromethyl)-N-(4-[[tris(propan-2-yl)silyl]oxy]phenyl)aniline
 2-methyl-3-[4-(6-trifluoromethyl-quinolin-2-yl)-piperazin-1-yl]-propionic acid 1-[(5-chloro-2,3-dihydro-1-benzofuran-2-yl)carbonyl]piperazine tert-butyl 4-[(5-chloro-2,3-dihydro-1-benzofuran-2-yl)carbonyl]piperazine-1-carboxylate (5-fluoro-2,3-dihydro-benzofuran-2-yl)-piperazin-1-yl-methanone
 4-(5-fluoro-2,3-dihydro-benzofuran-2-carbonyl)-piperazine-1-carboxylic acid tert-butyl ester 1-[[5-(trifluoromethyl)-2,3-dihydro-1-benzofuran-2-yl]methyl]piperazine 2-(iodomethyl)-5-(trifluoromethyl)-2,3-dihydro-1-benzofuran 2-chloro-1-[4-[(5-chloro-2,3-dihydro-1-benzofuran-2-yl)methyl]piperazin-1-yl]ethan-1-one
 1-[(5-chloro-2,3-dihydro-1-benzofuran-2-yl)methyl]piperazine 5-chloro-2-(chloromethyl)-2,3-dihydro-1-benzofuran 1-(5-fluoro-2,3-dihydro-benzofuran-2-ylmethyl)piperazine 5-fluoro-2-iodomethyl-2,3-dihydro-benzofuran
 2-(piperazin-1-yl)-6-(trifluoromethyl)quinoline N-[4-cyano-3-(trifluoromethyl)phenyl]piperidin-4-amine tert-butyl 4-[[4-cyano-3-(trifluoromethyl)phenyl]amino]piperidine-1-carboxylate 4-(4-cyano-3-trifluoromethyl-phenylamino)cyclohexanol
 (5S)-5-(aminomethyl)-3-(3-fluoro-4-morpholinophenyl)-1,3-oxazolidin-2-one methyl 4-(methylamino)-3-nitrobenzoate benzyl 5-indolecarboxylate 7-methyl-2-phenyl-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid ethyl ester
 2-methyl-benzothiazole-6-carboxylic acid 1-(2-chloroacetyl)thiazolidine 1-(methoxymethyl)indole-3-carboxylic acid methyl 5-methoxy-1-methyl-1H-indole-3-carboxylate
 methyl 1-methoxymethyl-1H-indole-3-carboxylate N,N,dimethyl-1,4-butanediamine 5-methoxy-2-[(4-methylphenyl)sulfonyl]isoindoline 3-Amino-1-(1,3-dihydroisoindol-2-yl)propan-1-one
 N-(2-aminoethyl)-2-quinolinecarboxamide 3-amino-1-(2,3-dihydroindol-1-yl)propan-1-one 7-methyl-2-phenyl-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid tert-butyl (3-(indolin-1-yl)-3-oxopropyl)carbamate
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