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 6-methyl-4-oxo-1,4-dihydro-pyridine-3-carboxylic acid hydrochloride tert-butyl 3-({4-chloro-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzoate 4-(4-chloro-5-(trifluoromethyl)pyrimidin-2-ylamino)-N-methylbenzamide (4-(4-chloro-5-(trifluoromethyl)pyrimidin-2-ylamino)phenyl)methanol
 N-(2-cyano-5-methyl-phenyl)-N-(methylsulfonyl)methanesulfonamide 4-(methanesulfonyl-methyl-amino)-2-methyl-pyrimidine-5-carboxylic acid amide N-(3-Aminomethyl-4-methyl-pyridin-2-yl)-N-methyl-methanesulfonamide N-(5-cyano-2-methyl-pyrimidin-4-yl)-N-methyl-methanesulfonamide
 N-(5-Cyano-2-methyl-pyridin-4-yl)-N-methyl-methanesulfonamide N-(6-chloro-2-cyano-pyridin-3-yl)-N-methyl-methanesulfonamide N-(2-cyano-5-methyl-phenyl)-methanesulfonamide N-(2-cyano-3-methyl-phenyl)-methanesulfonamide
 N-(3-cyano-4-methyl-phenyl)-N-methyl-methanesulfonamide N-(3-cyano-5-methyl-pyridin-2-yl)-N-methyl-methanesulfonamide N-(3-cyano-4-methyl-phenyl)-methanesulfonamide N-(3-cyano-6-methyl-pyridin-2-yl)-N-methyl-methanesulfonamide
 N-(3-cyano-4-methyl-pyridin-2-yl)-N-methyl-methanesulfonamide 1,4-dihydro-6-methyl-4-oxopyridine-3-carboxamide 6-methyl-4-oxo-1,4-dihydro-pyridine-3-carboxylic acid methyl ester 4-Bromo-1-(tert-butoxycarbonylamino)-7-[(methanesulfonyl)oxy]naphthalene
 (E)-8-(benzylideneamino)naphthalen-2-ol ethyl 1-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)cyclobutanecarboxylate 1-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)cyclobutanecarboxylic acid ethyl 3-(5-amino-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)propanoate
 tert-butyl 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)-2-methylpropanoate ethyl 2-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)-2-methylpropanoate ethyl 2-(5-amino-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)-2-methylpropanoate ethyl 3-(5-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-ylthio)propanoate
 tert-butyl 4-cyclopropylnaphthalen-1-ylcarbamate 1-amino-4-cyclopropylnaphthalene hydrochloride 1-amino-4-cyclopropylnaphthalene oxalate 2-Chlorobenzyl bromide
 3,4-dimethyl-1(2)H-pyrano[2,3-c]pyrazol-6-one 1-(4-chlorobenzyl)hydrazine Tri-tert-butylphosphonium Tetraphenylborate 4-((8-hydroxyquinolin-7-yl)(phenyl)methylamino)benzoic acid
 N-(5-(2,6-dimorpholinopyrimidin-4-yl)-4-(trifluoromethyl)pyridin-2-yl)acetamide 5-(2,6-dimorpholin-4-ylpyrimidin-4-yl)-4-trifluoromethylpyridin-2-ylamine hydrochloride 6-acetamido-4-(trifluoromethyl)pyridin-3-ylboronic acid 2-amino-4-chloroquinazoline
 5-(1H-Pyrazol-4-yl)-2-(6-((2,2,6,6-tetramethylpiperidin-4- yl)oxy)pyridazin-3-yl)phenol N-(5-bromo-4-(trifluoromethyl)pyridin-2-yl)acetamide 5-hydroxy-2-methylchromone 5-methoxy-2-methylchromone
 1-isopropyloxy-2-fluoro-4-bromobenzene N,N-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-hydroxy-6-methylphenyl)-2-phenylethanone 2-fluoro-N1,N1-dimethylbenzene-1,4-diamine
 N-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 2-(3-fluoro-4-isopropoxyphenyl)-4,4,5,5-tetramethyl-1,3,2- dioxaborolane 3-methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-1-indazole 4-bromo-2-fluoro-N,N-dimethylaniline
 5-amino-3-(piperidin-1-yl)-1H-pyrazole-4-carbonitrile 2-fluoro-N,N-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2-isopropoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrimidine 4-(4-bromo-2-fluorophenoxy)tetrahydro-2H-pyran
 3-morpholino-1H-pyrazolo[3,4-d]pyrimidin-4-amine 3-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 2-fluoro-N1-isopropylbenzene-1,4-diamine 3-(benzo[b]thiophen-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
 3-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 4-(3-iodo-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine tert-butyl 6-bromo-3-isopropyl-1H-indazole-1-carboxylate 4-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine
 3-iodo-N,N-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 3-bromo-5-methoxy-2-methyl-4H-chromen-4-one 3-iodo-N-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine N3,N3-dimethyl-1H-pyrazolo[3,4-d]pyrimidine-3,4-diamine
 3-ethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 2-fluoro-N-isopropyl-4-nitroaniline methyl 3-acetyl-1H-indole-6-carboxylate methyl 3-ethyl-1H-indole-6-carboxylate
 methyl 1-benzyl-1H-indole-6-carboxylate 1-phenyl-1,2,3-triazole-4-carboxylic acid 1-phenyl-1H-imidazole-4-carboxylic acid 1-(3-fluorophenyl)-1H-1,2,4-triazole-3-carboxylic acid
 1-(4-fluorophenyl)pyrazole-3-carboxylic acid ethyl 2-(4-hydroxypiperidin-1-yl)thiazole-4-carboxylate ethyl 1-(4-chlorophenyl)pyrazole-3-carboxylate (S)-tert-butyl 3-(6-chloroquinazoline-2-carboxamido)pyrrolidine-1-carboxylate
 (S)-tert-butyl N-(1-(pyrrolo[1,2-a]pyrazin-1-yl)pyrrolidin-3-yl)carbamate (S)-tert-butyl (1-(pyrazolo[1,5-a]pyrazin-4-yl)pyrrolidin-3-yl)carbamate (S)-tert-butyl (1-(imidazo[1,2-a]pyrazin-8-yl)pyrrolidin-3-yl)carbamate 1-o-tolyl-1H-pyrazole-3-carboxylic acid ethyl ester
 1-(tetrahydropyran-4-yl)-1H-pyrazole-3-carboxylic acid 5-isopropylpyrimidine-2-carboxylic acid ethyl 6-chloroquinazoline-2-carboxylate ethyl 2-(4-chloro-2-formylanilino)-2-oxoacetate
 6-methylquinazoline-2-carboxylic acid 4-chloropyrazolo[1,5-a]pyrazine 6-(4-hydroxypiperidin-1-yl)pyridazine-3-carboxylic acid methyl 6-(4-hydroxypiperidin-1-yl)pyridazine-3-carboxylate
 1-(4-fluorophenyl)-1,2,4-triazole-3-carbonyl chloride 1-(4-iodophenyl)-1,2,4-triazole-3-carboxylic acid methyl 1-(4-iodophenyl)-1,2,4-triazole-3-carboxylate 1-chloro-3-isopropylpyrrolo[1,2-a]pyrazine
 3-isopropylpyrrolo[1,2-a]pyrazin-1(2H)-one 1-chloro-3-ethylpyrrolo[1,2-a]pyrazine 3-ethylpyrrolo[1,2-a]pyrazin-1(2H)-one 1-(o-tolyl)pyrazole-3-carboxylic acid
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